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382 items
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Overcoming the Low Oral Bioavailability of Deuterated Pyrazoloquinolinone Ligand DK-I-60-3 by Nanonization: A Knowledge-Based Approach
Jelena R. Mitrović , Branka Divović-Matović, Daniel E. Knutson, Jelena B. Ðoković, Aleksandar Kremenović, Vladimir D. Dobričić, Danijela V. Randjelović, Ivana Pantelić, James M. Cook, Miroslav M. Savić, Snežana D. Savić (2021)Poor water solubility of new chemical entities is considered as one of the main obstacles in drug development, as it usually leads to low bioavailability after administration. To overcome these problems, the selection of the appropriate formulation technology needs to be based on the physicochemical properties of the drug and introduced in the early stages of drug research. One example of the new potential drug substance with poor solubility is DK-I-60-3, deuterated pyrazoloquinolinone, designed for the treatment of various neuropsychiatric ...Jelena R. Mitrović , Branka Divović-Matović, Daniel E. Knutson, Jelena B. Ðoković, Aleksandar Kremenović, Vladimir D. Dobričić, Danijela V. Randjelović, Ivana Pantelić, James M. Cook, Miroslav M. Savić, Snežana D. Savić. "Overcoming the Low Oral Bioavailability of Deuterated Pyrazoloquinolinone Ligand DK-I-60-3 by Nanonization: A Knowledge-Based Approach" in Pharmaceutics, MDPI, Basel, Switzerland (2021). https://doi.org/10.3390/pharmaceutics13081188
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Numerical modelling of a single intra-oceanic subduction for the origin of the Balkan ophiolites
Nikola Stanković, Vesna Cvetkov, Vladica Cvetković. "Numerical modelling of a single intra-oceanic subduction for the origin of the Balkan ophiolites" in 5th Congress Geologists of the Republic of North Macedonia, Ohrid, 28-29. 10. 2024, Македонско геолошко друштво (2024)
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Structural and microstructural study of brookite based TiO2 nanocomposites with carbon black (C)
Structural and microstructural properties of TiO2-based nanocomposites with carbon black (C), synthesized by sol-gel-hydrothermal method, have been studied by XRPD and Raman scattering. Detailed size-strain analyses of XRPD and Raman scattering results are presented in order to investigate the influence of C content on brokite and anatase phase formation. The XRPD size-strain analyses have resulted in reliable structure and microstructure results for both anatase and brookite and their relative abundance ratio has been refined by Rietveld method. The brookite ...Aleksandar Kremenović, Mirjana Grujić-Brojčin, Nataša Tomić, Maja Šćepanović. "Structural and microstructural study of brookite based TiO2 nanocomposites with carbon black (C)" in The European Powder Diffraction Conference (EPDIC) Book of Abstracts, Šibenik, 31 May - 3 June 2022, EPDIC (2022)
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Effect of natural gas composition on methane number: A case of gas reservoirs in Serbia
Natural gas is considered as the most environmentally acceptable fossil fuel, thus it is an alternative to petroleum derivate, dominantly used in internal combustion engines. Physical properties of a fuel as well as behavior during combustion process are affected by its composition. This article presents analysis of effect of natural gas composition on methane number (MN), conducted for natural gas deposits in Serbia. For empirically determination of MN: California air resources board (CARB) method and Linear and Anstalt für ...Marija Živković, Milica Ivić, Dejan Ivezić, Aleksandar Madžarević. "Effect of natural gas composition on methane number: A case of gas reservoirs in Serbia" in Energy Sources, Part A: Recovery, Utilization, and Environmental Effects (2017). https://doi.org/10.1080/15567036.2017.1403518
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Развој геолошког терминолошког речника ГеолИССТерм
Ranka Stanković, Branislav Trivić, Olivera Kitanović, Branislav Blagojević, Velizar Nikolić. "Развој геолошког терминолошког речника ГеолИССТерм" in INFOteka: časopis za informatiku i bibliotekarstvo, Beograd : Zajednica biblioteka univerziteta u Srbiji (2011)
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The influence of structural modification of Pd(II) pincer-type complexes on the kinetics of substitution reactions
Snežana Jovanović Stević, Snežana Radisavljević, Aleksandar Mijatović, Biljana Petrović, Ana Kesić (2023)This mini-review summarizes the kinetic data obtained for the substitution reactions of some palladium(II) complexes containing bis-pyrazolylpyridine derivatives as pincer-type ligands with biologically significant nitrogen- and sulfur-donor biomolecules as nucleophiles. Three structurally different palladium(II) complexes were selected: [Pd(L1)Cl]+ (Pd1), [Pd(L2)Cl]+ (Pd2) and [Pd(L3)Cl]+ (Pd3) (where L1 = bis(2-(1H-pyrazol-1-yl)ethyl)amine, L2 = 2,6-bis(5-(tert-butyl)-1H-pyrazol-3-yl)pyridine, and L3 = 2,6-bis(5-(tert-butyl)-1-methyl-1H-pyrazol-3-yl)pyridine, while for the entering nucleophiles were used thiourea (Tu), L-methionine (L-met), and guanosine-5’-monophosphate (5’-GMP). Kinetic measurements were carried out for all systems as pseudo-first ...Snežana Jovanović Stević, Snežana Radisavljević, Aleksandar Mijatović, Biljana Petrović, Ana Kesić. "The influence of structural modification of Pd(II) pincer-type complexes on the kinetics of substitution reactions" in 2nd International Conference on Chemo and BioInformatics ICCBIKG 2023, 28-29 September 2023, Institute for Information Technologies, University of Kragujevac, Serbia, Kragujevac : Institute for Information Technologies, University of Kragujevac (2023)
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Constitutive Model for Analysis of Long-Term Municipal Solid Waste Landfill Settlement
Irena Basarić Ikodinović, Dragoslav Rakić, Mirjana Vukićević, Sanja Jocković, Jovana Janković Pantić (2022)Large long-term settlement occurs at the municipal solid waste landfills over an extended period of time which may lead to breakage of the geomembrane, damage of the cover systems, other protective systems or facilities constructed on top of a landfill. Also, municipal solid waste is an extremely heterogeneous material and its properties vary over location and time within a landfill. These material characteristics require the formulation of a new constitutive model to predict the long-term settlement of municipal solid ...Irena Basarić Ikodinović, Dragoslav Rakić, Mirjana Vukićević, Sanja Jocković, Jovana Janković Pantić. "Constitutive Model for Analysis of Long-Term Municipal Solid Waste Landfill Settlement" in ICEG 2022: International Conference on Environmental Geotechnics, World Academy of Science, Engineering and Technology (2022)
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Human Hemoglobin and Antipsychotics Clozapine, Ziprasidone and Sertindole: Friends or Foes?
Lena Platanić Arizanović, Nikola Gligorijević, Ilija Cvijetić, Aleksandar Mijatović, Maja Krstić Ristivojević, Simeon Minić, Aleksandra Nikolić Kokić, Čedo Miljević, Milan Nikolić (2023)Packed with hemoglobin, an essential protein for oxygen transport, human erythrocytes are a suitable model system for testing the pleiotropic effects of lipophilic drugs. Our study investi gated the interaction between antipsychotic drugs clozapine, ziprasidone, sertindole, and human hemoglobin under simulated physiological conditions. Analysis of protein fluorescence quenching at different temperatures and data obtained from the van’t Hoff diagram and molecular docking indicate that the interactions are static and that the tetrameric human hemoglobin has one binding site for ...Inorganic Chemistry, Organic Chemistry, Physical and Theoretical Chemistry, Computer Science Applications, Spectroscopy, Molecular Biology, General Medicine, CatalysisLena Platanić Arizanović, Nikola Gligorijević, Ilija Cvijetić, Aleksandar Mijatović, Maja Krstić Ristivojević, Simeon Minić, Aleksandra Nikolić Kokić, Čedo Miljević, Milan Nikolić. "Human Hemoglobin and Antipsychotics Clozapine, Ziprasidone and Sertindole: Friends or Foes?" in International Journal of Molecular Sciences, MDPI AG (2023). https://doi.org/10.3390/ijms24108921
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LRMI markup of OER content within the BAEKTEL project
Ranka Stanković, Daniela Carlucci, Olivera Kitanović, Nikola Vulović, Bojan Zlatić. "LRMI markup of OER content within the BAEKTEL project" in The Sixth International Conference on e-Learning (eLearning-2015), September 2015, Belgrade, Serbia, Belgrade : Belgrade Metropolitan Univesity (2015)
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Some examples of interactions between certain rare earth elements and soil
Zlatko Nikolovski, Jelena Isailović, Dejan Jeremić, Sabina Kovač, Ilija Brčeski. "Some examples of interactions between certain rare earth elements and soil" in Journal of the Serbian Chemical Society, National Library of Serbia (2021). https://doi.org/10.2298/JSC211006095N
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Solid state synthesis of extra phase-pure Li4Ti5O12 spinel
Фазно чист спинел Li4Ti5O12 са величином честица мањом од 500 nm добијен је реакцијом у чврстом стању из стехиометријске смеше наноанатаса (ТiО2) и Li2CO3 која је претходно активирана механохемијским поступком. Реакција у чврстом стању у потпуности се завршава за само 4 часа на температури од 800 ºC. Уз помоћ XRPD, SEM и TG/DSC анализе испитане су структурне и микроструктурне карактеристике добијеног спинела, механизам реакције између анатаса и Li2CO3, као и термичка стабилност Li4Ti5O12. Реакција започиње разлагањем Li2CO3 на температурама ...дифракција рендгенских зрака, механизам реакције, термичка стабилност, Li4Ti5O12, спинел, фазно чист узоракIvana Veljković, Dejan Poleti, Ljiljana Karanović, Miodrag Zdujić, Goran Branković. "Solid state synthesis of extra phase-pure Li4Ti5O12 spinel" in Science of Sintering, National Library of Serbia (2011). https://doi.org/10.2298/SOS1103343V
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A proposal for the landslide damage questionnaire in suburban areas
Landslides are one of the most often natural disasters that have an extensive impact on society including loss of life, destruction of infrastructure and properties, damage to land and loss of natural resources. Landslide losses can significantly vary and they depend on a variety of different criteria such as the size and type of landslide, lithological setting of terrain, the terrain slope gradient, the quality of materials used for construction, and the construction typology. Damage from landslides is usually ...Uroš Đurić, Biljana Abolmasov, Miloš S. Marjanović, Sanja Jocković, Miloš D. Marjanović. "A proposal for the landslide damage questionnaire in suburban areas " in 5th Regional symposium on landslides in Adriatic–Balkan Region, 23-26 March 2022, Faculty of Civil Engineering, University of Rijeka and Faculty of Mining, Geology and Petroleum Engineering, University of Zagreb (2022)
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Unusually sluggish microemulsion system with water, toluene and a technical branched alkyl polyethoxylate
Marija Ilić, Franz-Hubert Haegel, Vesna Pavelkić, Snežana Zlatanović, Zoran Marković, Aleksandar Cvjetić (2015)Microemulsion systems with water, toluene and nonionic surfactants are interesting for application due to the excellent solvent properties of aromatic hydrocarbons. In this study, the pseudo-binary phase diagram (“fish-diagram”) of such a ternary system was investigated using a branched technical alkyl polyethoxylate. Lutensol ON 50 (i-C10E5) was considered a suitable surfactant. The system with technical branched i-C10E5 exhibits very long, and for compositions near optimum solubilization, i.e., the minimum content of surfactant needed for a bicontinuous microemulsion, extremely long ...микроемулзија, толуен, оксоалкохол етоксилат, термодинамичка стабилност, тернарни фазни дијаграми, дијаграми „fish“Marija Ilić, Franz-Hubert Haegel, Vesna Pavelkić, Snežana Zlatanović, Zoran Marković, Aleksandar Cvjetić. "Unusually sluggish microemulsion system with water, toluene and a technical branched alkyl polyethoxylate" in Chemical Industry and Chemical Engineering Quarterly (2015). https://doi.org/10.2298/CICEQ141012045I
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Correlation Between Dynamic CBR and Compaction and Bearing Capacity of Pavement Foundation Layers
This paper presents a dynamic California Bearing Ratio (CBRd) device that can be used on a prepared pavement foundation layer to obtain a certain parameter of the tested material in the laboratory and in situ in a direct and fast way. For the selected natural material (gravel), it is shown that the laboratory CBRd can be used to estimate the compaction and bearing capacity, because it correlates well with the parameters of the standard and modifed Proctor compaction tests. ...korelacija parametara, donji slojevi saobraćajnica, laboratorijska i terenska ispitivanja, dinamički kalifornijski indeks nosivosti CBRd... pavement is built (up- per bearing layers and asphalt and concrete layers). The contributions of this study are as follows: – the geotechnical properties of the selected material (gravel) were determined, and the physical-me- chanical parameters are defined based on laboratory testing for incorporation ...
... has been presented [5], and the correlations of the parameters of the laboratory dynamic California Bearing Ratio (CBR, ) with the com- paction properties of sandy soil have been reported [4]. Owing to its short duration and ease, CBR, testing using a LWD can become widespread as an alterna- tive ...
... optimal water content w„„i (SP) = 9.5% and Wopt (MP) = 8.6%. The CBR,, SPLT, and LWD were used to estimate the compaction and bearing capacity properties of the selected natural material (gravel) embedded in the final layer of the substrate (subgrade). CBR;y is a complex measure of the strength ...Milan Bogdanović, Snežana Bogdanović, Dragoslav Rakić, Irena Basarić Ikodinović. "Correlation Between Dynamic CBR and Compaction and Bearing Capacity of Pavement Foundation Layers" in Soil Mechanics and Foundation Engineering, Springer Science and Business Media LLC (2024). https://doi.org/10.1007/s11204-024-09939-x
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WS4LR - a Worksation for Lexical Resources
Cvetana Krstev, Ranka Stanković, Duško Vitas, Ivan Obradović. "WS4LR - a Worksation for Lexical Resources" in Proceedings of the Fifth Interantional Conference on Language Resources and Evaluation, Genoa, Italy, May 2006, ELRA - European Language Resources Association (2006)
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Some models for determination of parameters of the soil oscillation law during blasting operations
Suzana Lutovac, Dragan Medenica, Branko Gluščević, Rade Tokalić, Čedomir Beljić. "Some models for determination of parameters of the soil oscillation law during blasting operations" in Energies, Basel, Switzerland : MDPI (2018). https://doi.org/10.3390/en9080617
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Development of a petrographic classification system for organic particles affected by self-heating in coal waste. (An ICCP Classification System, Self-heating Working Group – Commission III)
M. Misz-Kennan, J. Kus, D. Flores, C. Avila, Z. Büçkün, N. Choudhury, K. Christanis, J.P. Joubert, S. Kalaitzidis, A.I. Karayigit, M. Malecha, M. Marques, P. Martizzi, J.M.K. O'Keefe, W. Pickel, G. Predeanu, S. Pusz, J. Ribeiro, S. Rodrigues, A.K. Singh, I. Suárez-Ruiz, I. Sýkorová, N.J. Wagner, D. Životić (2020)Self-heating of coal waste is a major problem in the leading coal-producing and consuming countries, independent of the recent or past coal exploitation history. The phenomenon of self-heating is dependent on many factors such as the properties of organic matter (maceral composition and rank), moisture and pyrite content, climate effects, and storage conditions (shape of the dump or compaction of the coal waste). Once deposited, coal waste undergoes oxidation, which can lead to self- heating with the overall temperatures ...... n criteria were nu- merous and included among others an appropriate hierarchical struc- ture by optical appearance (e.g., physical properties) and/or optical properties, grouping relevant categories and sub-categories as well as valid annotation types. Thus, the comparison of data sets based on former ...
... countries, in- dependent of the recent or past coal exploitation history. The phenomenon of self-heating is dependent on many factors such as the properties of organic matter (maceral composition and rank), moisture and pyrite content, climate effects, and storage conditions (shape of the dump or compaction ...
... 2020.103411 mailto:magdalena.misz@us.edu.pl bitumen, chars, graphite, and coke). Altered particles were further divided according to their optical properties (porous, massive; isotropic, anisotropic). For altered particles the following specific features were distinguished: fractures, fissures, cracks; ...M. Misz-Kennan, J. Kus, D. Flores, C. Avila, Z. Büçkün, N. Choudhury, K. Christanis, J.P. Joubert, S. Kalaitzidis, A.I. Karayigit, M. Malecha, M. Marques, P. Martizzi, J.M.K. O'Keefe, W. Pickel, G. Predeanu, S. Pusz, J. Ribeiro, S. Rodrigues, A.K. Singh, I. Suárez-Ruiz, I. Sýkorová, N.J. Wagner, D. Životić. "Development of a petrographic classification system for organic particles affected by self-heating in coal waste. (An ICCP Classification System, Self-heating Working Group – Commission III)" in International Journal of Coal Geology, Elsevier BV (2020). https://doi.org/10.1016/j.coal.2020.103411
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A survey of greenhouse gases production in central European lignites
Anna Pytlak, Anna Szafranek-Nakonieczna, Weronika Goraj, Izabela Śnieżyńska, Aleksandra Krążała, Artur Banach, Ivica Ristović, Mirosław Słowakiewicz, Zofia Stępniewska (2021)Anna Pytlak, Anna Szafranek-Nakonieczna, Weronika Goraj, Izabela Śnieżyńska, Aleksandra Krążała, Artur Banach, Ivica Ristović, Mirosław Słowakiewicz, Zofia Stępniewska. "A survey of greenhouse gases production in central European lignites" in Science of The Total Environment, Elsevier (2021). https://doi.org/10.1016/j.scitotenv.2021.149551
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Groundwater as an important resources in emergency situations of the Republic of Serbia
Boris Vakanjac, Radoje Banković, Vesna Ristić-Vakanjac, Saša Milanović, Ljiljana Vasić, Saša Bakrač, Nikola Kozić (2024)Groundwater is a renewable resource wholly or partially protected from external influences (pollutants) by nature. Currently, about 75% of the population of the Republic of Serbia meets its water needs by using underground water. Hence, this water represents an essential strategic resource of our country; according to data from the Water Management Foundation of the Republic of Serbia (VOS, 2001), water from existing sources is used in quantities of about 23 m3/s. As 67.13 m3/s is the estimated potential ...Boris Vakanjac, Radoje Banković, Vesna Ristić-Vakanjac, Saša Milanović, Ljiljana Vasić, Saša Bakrač, Nikola Kozić. "Groundwater as an important resources in emergency situations of the Republic of Serbia" in 11th International Scientific Conference on Defensive Technologies - OTEX 2024, Tara, October 2024, Military Technical Institute, Belgrade (2024). https://doi.org/10.5937/OTEH24122V
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Synthesis, characterization, biomolecular interactions, molecular docking, and in vitro and in vivo anticancer activities of novel ruthenium(III) Schiff base complexes
Milica Međedović, Aleksandar Mijatović, Rada Baošić, Dejan Lazić, Žiko Milanović, Zoran Marković, Jelena Milovanović, Dragana Arsenijević, Bojana Stojanović, Miloš Arsenijević, Marija Milovanović, Biljana Petrović, Ana Rilak Simović (2023)In order to discover new anticancer drugs, novel ruthenium(III) complexes [Ru(L)Cl(H2O)], where L is tetradentate Schiff base bis(acetylacetone)ethylendiimine (acacen, 1), bis(benzoylacetone)ethylendiimine (bzacen, 2), (acetylacetone)(benzoylaceton)ethylendiimine (acacbzacen, 3), bis(acetylacetone)propylendiimine (acacpn, 4), bis(benzoylacetone)propylendiimine (bzacpn, 5) or (acetylacetone)(benzoylaceton)propylendiimine (acacbzacpn, 6), were synthesized. The complexes 1 – 6 were characterized by elemental analysis, molar conductometry, and by various spectroscopic techniques, such as UV–Vis, IR, EPR, and ESI-MS. Based on in vitro DNA/BSA experiments, complexes 2 (bzacen) and 5 (bzacpn) with two aromatic rings showed ...Milica Međedović, Aleksandar Mijatović, Rada Baošić, Dejan Lazić, Žiko Milanović, Zoran Marković, Jelena Milovanović, Dragana Arsenijević, Bojana Stojanović, Miloš Arsenijević, Marija Milovanović, Biljana Petrović, Ana Rilak Simović. "Synthesis, characterization, biomolecular interactions, molecular docking, and in vitro and in vivo anticancer activities of novel ruthenium(III) Schiff base complexes" in Journal of Inorganic Biochemistry, Elsevier BV (2023). https://doi.org/10.1016/j.jinorgbio.2023.112363